BDBM253656 US9458201, 146

SMILES CC(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H]1CCCC(=O)NCC[C@H](NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H]2C[C@@H](O)CN2C1=O)C(O)=O

InChI Key InChIKey=NGRHUDDGBSABPT-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 253656   

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandPNGBDBM253656(US9458201, 146)
Affinity DataKi:  3nM ΔG°:  -12.1kcal/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
Go to US Patent