BDBM246317 US9434693, 11

SMILES COc1ccccc1-n1nc(O[C@@H]2CC[C@@H](CC2)NC(=O)OC(C)(C)C)cc1-c1ccc(Cl)cc1

InChI Key InChIKey=XNUZTIQWJMXUHN-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 246317   

TargetVoltage-dependent L-type calcium channel subunit beta-3/N-type calcium channel subunit alpha-1B/calcium channel subunit alpha-2/delta-1(Human)
Janssen Pharmaceutica

US Patent

LigandBDBM246317(US9434693, 11)Copy SMILESCopy InChI

Affinity DataIC50: 62nMAssay Description:Calcium mobilization responses to KCl depolarization were evaluated by measuring the intensity of calcium-mediated fluorescent signal in the presence...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/28/2017
Entry Details
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