BDBM24397 2-chloro-N-[(3S)-1-[(2R)-2,3-dihydroxypropyl]-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]-6H-thieno[2,3-b]pyrrole-5-carboxamide::3,4-dihydro-2-quinolone (DHQ) derivative, 36

SMILES OC[C@H](O)CN1C(=O)[C@H](Cc2ccccc12)NC(=O)c1cc2cc(Cl)sc2[nH]1

InChI Key InChIKey=UICNBXVDHCBKCE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 24397   

TargetGlycogen phosphorylase, liver form(Human)
Astrazeneca

LigandPNGBDBM24397(2-chloro-N-[(3S)-1-[(2R)-2,3-dihydroxypropyl]-2-ox...)
Affinity DataIC50: 27nMAssay Description:The inhibitory activity of the test compounds against human recombinant glycogen phosphorylase a (GPa) was monitored using 96-well microplate format....More data for this Ligand-Target Pair
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Date in BDB:
9/15/2008
Entry Details Article
PubMed