BDBM240792 H-D-Ser-homoPhe-Arg-OH (3)

SMILES N[C@H](CO)C(=O)N[C@H](CCc1ccccc1)C(=O)N[C@H](CCCNC(N)=N)C(O)=O

InChI Key InChIKey=ISXAPWUOYYNLBV-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 240792   

TargetPlasminogen(Human)
Medical University of Bialystok

LigandPNGBDBM240792(H-D-Ser-homoPhe-Arg-OH (3))
Affinity DataKi:  5.90E+3nMpH: 7.4Assay Description:Buffer and 0.1 mL of enzyme solution was added to 0.2 mL of examined compounddissolved in 0.15 M NaCl (as control 0.15 M NaCl). The buffer and the en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetProthrombin(Human)
Medical University of Bialystok

LigandPNGBDBM240792(H-D-Ser-homoPhe-Arg-OH (3))
Affinity DataKi:  1.61E+4nMpH: 8.4Assay Description:Buffer and 0.1 mL of enzyme solution was added to 0.2 mL of examined compounddissolved in 0.15 M NaCl (as control 0.15 M NaCl). The buffer and the en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Medical University of Bialystok

LigandPNGBDBM240792(H-D-Ser-homoPhe-Arg-OH (3))
Affinity DataKi:  2.39E+4nMpH: 7.5Assay Description:Buffer and 0.1 mL of enzyme solution was added to 0.2 mL of examined compounddissolved in 0.15 M NaCl (as control 0.15 M NaCl). The buffer and the en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Medical University of Bialystok

LigandPNGBDBM240792(H-D-Ser-homoPhe-Arg-OH (3))
Affinity DataKi:  5.66E+5nMpH: 8.8Assay Description:Buffer and 0.1 mL of enzyme solution was added to 0.2 mL of examined compounddissolved in 0.15 M NaCl (as control 0.15 M NaCl). The buffer and the en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed