BDBM240742 US9422263, 43::US9422263, 44

SMILES CN1C(C)=C(C#N)C(C(C#N)=C1C(F)(F)F)c1ccc2[nH]nc(C)c2c1

InChI Key InChIKey=JVLIJULZEKHEPQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 240742   

TargetHepatocyte growth factor receptor(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM240742(US9422263, 44 | US9422263, 43)
Affinity DataIC50: 9nMpH: 7.0 T: 2°CAssay Description:Recombinant human c-Met protein (Invitrogen, Carlsbad, Calif., USA) is used. As substrate for the kinase reaction the peptide KKKSPGEYVNIEFG (JPT, Ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
Go to US Patent

TargetHepatocyte growth factor receptor(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM240742(US9422263, 44 | US9422263, 43)
Affinity DataIC50: 8nMpH: 7.0 T: 2°CAssay Description:Recombinant human c-Met protein (Invitrogen, Carlsbad, Calif., USA) is used. As substrate for the kinase reaction the peptide KKKSPGEYVNIEFG (JPT, Ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
Go to US Patent