BDBM236399 US9365576, 152
SMILES CNc1ncc(-c2cc3C(=O)N(C(c3n2C(C)C)c2ccc(Cl)cc2)c2c[nH]c(=O)c(Cl)c2)c(OC)n1
InChI Key InChIKey=XBYKCKQFYADHRG-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 236399
TargetCellular tumor antigen p53 [18-26]/E3 ubiquitin-protein ligase Mdm2 [2-188](Human)
Novartis
US Patent
Novartis
US Patent
Affinity DataIC50: 0.166nMT: 2°CAssay Description:Assay 2: The test is performed in white 384-well plates (Greiner Bio-One, reference 781207) in a total volume of 60 μL by adding 1 μL of compou...More data for this Ligand-Target Pair