BDBM230879 US9346822, 41

SMILES CCOCCN(C)Cc1c(sc2n(Cc3c(F)cccc3F)c(=O)n(-c3ccccn3)c(=O)c12)-c1ccc(NC(=O)NOC)cc1

InChI Key InChIKey=MNXSZYSLNRUFIA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 230879   

TargetGonadotropin-releasing hormone receptor(Human)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM230879(US9346822, 41)
Affinity DataIC50: 0.100nMAssay Description:The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2017
Entry Details
Go to US Patent

TargetGonadotropin-releasing hormone receptor(Crab-eating macaque)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM230879(US9346822, 41)
Affinity DataIC50: 3nMAssay Description:The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2017
Entry Details
Go to US Patent