BDBM229678 US9334269, 5

SMILES CNC(=O)c1cccc(Nc2ncnc(n2)N2CC(COc3ccc(cc3)C(F)(F)F)C2)c1

InChI Key InChIKey=XKJSUDVVZHDZIZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 229678   

TargetSodium channel protein type 9 subunit alpha(Human)
Amgen

US Patent

LigandBDBM229678(US9334269, 5)Copy SMILESCopy InChI

Affinity DataIC50: 200nMAssay Description:Compounds were tested on human Nav1.7 (hNav1.7) expressed stably in 293 cells, which have no endogenous sodium channels. Two forms of whole-cell patc...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
5/31/2017
Entry Details
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