BDBM228845 FITC-LQEEWETVM::FITC-PTHRct9

SMILES CSCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=S)Nc1ccc2c(c1)C(=O)OC21c2ccc(O)cc2Oc2cc(O)ccc12)[C@@H](C)O)C(C)C)C(O)=O

InChI Key InChIKey=YAHDCUGORQRYOK-UHFFFAOYSA-N

Data  8 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 228845   

TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Human)
The University of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  400nMpH: 6.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Human)
The University of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  400nMpH: 6.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Human)
The University of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  1.00E+3nMpH: 7.0 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Human)
The University of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  600nMpH: 7.0 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Human)
The University of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  1.00E+3nMpH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Human)
The University of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  600nMpH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [1-140](Human)
The University of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  4.70E+3nMpH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Human)
The University of Queensland

LigandPNGBDBM228845(FITC-LQEEWETVM | FITC-PTHRct9)
Affinity DataKd:  2.40E+3nMpH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed