BDBM22198 1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(2-phenylethyl)piperazine::CHEMBL26649::GBR 12935 Analogue, 38

SMILES Fc1ccc(cc1)C(OCCN1CCN(CCc2ccccc2)CC1)c1ccc(F)cc1

InChI Key InChIKey=AASZEODWFQQIRF-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 22198   

TargetSodium-dependent dopamine transporter(Rat)
National Taiwan University

LigandPNGBDBM22198(CHEMBL26649 | 1-{2-[bis(4-fluorophenyl)methoxy]eth...)
Affinity DataKi:  8nMAssay Description:The assay was initiated by the addition of membranes to binding buffer containing test compound, blocker, and radioligand. The samples were incubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2008
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
National Taiwan University

LigandPNGBDBM22198(CHEMBL26649 | 1-{2-[bis(4-fluorophenyl)methoxy]eth...)
Affinity DataKi:  8nMAssay Description:Binding affinity for dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Taiwan University

LigandPNGBDBM22198(CHEMBL26649 | 1-{2-[bis(4-fluorophenyl)methoxy]eth...)
Affinity DataKi:  36nMAssay Description:The assay was initiated by the addition of membranes to binding buffer containing test compound, blocker, and radioligand. The samples were incubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2008
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
National Taiwan University

LigandPNGBDBM22198(CHEMBL26649 | 1-{2-[bis(4-fluorophenyl)methoxy]eth...)
Affinity DataKi:  36nMAssay Description:Binding affinity for serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed