BDBM22144 aza-peptide Michael acceptor, 5x::benzyl N-[(1S)-1-{[(2S)-1-[(2E)-3-[N-(carbamoylmethyl)hydrazido]-N-methyl-N-{1-[methyl(2-phenylethyl)carbamoyl]-2-phenylethyl}prop-2-enamide]-1-oxopropan-2-yl]carbamoyl}ethyl]carbamate
SMILES C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)C(=O)NN(CC(N)=O)C(=O)C=CC(=O)N(C)C(Cc1ccccc1)C(=O)N(C)CCc1ccccc1
InChI Key InChIKey=AQPJVUBLQGYXRV-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 22144
Affinity DataIC50: 750nMT: 2°CAssay Description:AE activity in the induction medium was measured with the substrate Cbz-Ala-Ala-Asn-AMC. In a black 96-well microtiter plate, aza-peptidyl inhibitors...More data for this Ligand-Target Pair
TargetClan CD, family C13, asparaginyl endopeptidase-like cysteine peptidase(Trichomonas vaginalis G3)
Georgia Institute of Technology
Georgia Institute of Technology
Affinity DataIC50: 80nMT: 2°CAssay Description:AE activity in the induction medium was measured with the substrate Cbz-Ala-Ala-Asn-AMC. In a black 96-well microtiter plate, aza-peptidyl inhibitors...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMT: 2°CAssay Description:AE activity in the induction medium was measured with the substrate Cbz-Ala-Ala-Asn-AMC. In a black 96-well microtiter plate, aza-peptidyl inhibitors...More data for this Ligand-Target Pair