BDBM213821 US9296775, 1

SMILES CC(C)c1[nH]nc(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)c1Cc1ccc(\C=C\CCN2CCCC3(CCNCC3)C2)cc1C

InChI Key InChIKey=LVPGRGRCROHTBW-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 213821   

TargetSodium/glucose cotransporter 1(Human)
Eli Lilly

US Patent
LigandPNGBDBM213821(US9296775, 1)
Affinity DataIC50: 26nMpH: 7.5 T: 2°CAssay Description:The SGLT activity is measured as sodium-dependent 14C-AMG uptake in the above cell lines described as follows. One hundred uL of culture medium conta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2017
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Eli Lilly

US Patent
LigandPNGBDBM213821(US9296775, 1)
Affinity DataIC50: 6.10E+3nMpH: 7.5 T: 2°CAssay Description:The SGLT activity is measured as sodium-dependent 14C-AMG uptake in the above cell lines described as follows. One hundred uL of culture medium conta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2017
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase Sgk1(Mouse)
Eli Lilly

US Patent
LigandPNGBDBM213821(US9296775, 1)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The SGLT activity is measured as sodium-dependent 14C-AMG uptake in the above cell lines described as follows. One hundred uL of culture medium conta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2017
Entry Details
Go to US Patent