BDBM213771 US9284302, 1

SMILES Cc1nc(C)n(n1)-c1cc(nc(C)n1)C1(O)CC(C1)c1nc2ccccc2n1C

InChI Key InChIKey=ZGVBVZBTPMOZPJ-UHFFFAOYSA-N

Data  1 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 213771   

TargetIsoform PDE10A2 of cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A (PDE10A2)(Human)
Merck Sharp & Dohme

US Patent

LigandBDBM213771(US9284302, 1)Copy SMILESCopy InChI

Affinity DataKi: >75nMAssay Description:In a typical experiment the PDE10 inhibitory activity of the compounds of the present invention was determined in accordance with the following exper...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
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Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/21/2017
Entry Details
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