BDBM20409 3-1H-indazol-4-yl-1-[(1R)-1-(naphthalen-2-yl)ethyl]urea::indazole antagonist, (R)-16c

SMILES C[C@@H](NC(=O)Nc1cccc2[nH]ncc12)c1ccc2ccccc2c1

InChI Key InChIKey=ZMOPUGNHDAYKSY-UHFFFAOYSA-N

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20409   

LigandPNGBDBM20409(3-1H-indazol-4-yl-1-[(1R)-1-(naphthalen-2-yl)ethyl...)
Affinity DataEC50:  123nMpH: 7.4 T: 2°CAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2008
Entry Details Article
PubMed