BDBM20375 1-[(1-ethyl-2,3-dihydro-1H-indol-5-yl)methyl]-3-(1-methyl-1H-indazol-4-yl)urea::Indazole Analogue, 69

SMILES CCN1CCc2cc(CNC(=O)Nc3cccc4n(C)ncc34)ccc12

InChI Key InChIKey=GOZSIGIHYMBLDA-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20375   

LigandPNGBDBM20375(1-[(1-ethyl-2,3-dihydro-1H-indol-5-yl)methyl]-3-(1...)
Affinity DataEC50:  305nMAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2008
Entry Details Article
PubMed