BDBM20374 1-[(1-ethyl-2,3-dihydro-1H-indol-5-yl)methyl]-3-1H-indazol-4-ylurea::Indazole Analogue, 68

SMILES CCN1CCc2cc(CNC(=O)Nc3cccc4[nH]ncc34)ccc12

InChI Key InChIKey=CLIRFEGEDUGTMQ-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20374   

LigandPNGBDBM20374(1-[(1-ethyl-2,3-dihydro-1H-indol-5-yl)methyl]-3-1H...)
Affinity DataEC50:  285nMAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2008
Entry Details Article
PubMed