BDBM20372 1-({2,5-difluoro-4-[(1R,5S)-3-oxo-8-azabicyclo[3.2.1]octan-8-yl]phenyl}methyl)-3-1H-indazol-4-ylurea::Indazole Analogue, 66

SMILES Fc1cc(N2[C@H]3CC[C@@H]2CC(=O)C3)c(F)cc1CNC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=CLRSHLSJDZBRGM-UHFFFAOYSA-N

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20372   

LigandPNGBDBM20372(1-({2,5-difluoro-4-[(1R,5S)-3-oxo-8-azabicyclo[3.2...)
Affinity DataEC50:  157nMAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2008
Entry Details Article
PubMed