BDBM20368 1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3,5-difluorophenyl}methyl)-3-1H-indazol-4-ylurea::Indazole Analogue, 62

SMILES Fc1cc(CNC(=O)Nc2cccc3[nH]ncc23)cc(F)c1N1[C@H]2CC[C@@H]1CCC2

InChI Key

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20368   

LigandPNGBDBM20368(1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3,5-...)
Affinity DataEC50:  12.6nMAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2008
Entry Details Article
PubMed