BDBM20363 1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2-(trifluoromethyl)phenyl}methyl)-3-1H-indazol-4-ylurea::Indazole Analogue, 57

SMILES FC(F)(F)c1cc(ccc1CNC(=O)Nc1cccc2[nH]ncc12)N1[C@H]2CC[C@@H]1CCC2

InChI Key

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20363   

LigandPNGBDBM20363(1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2-(t...)
Affinity DataEC50:  54.5nMpH: 7.4 T: 2°CAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2008
Entry Details Article
PubMed