BDBM202418 US9238644, 24A

SMILES CC(N)c1ccc(Nc2ncc(Cl)c(CCc3ccccc3C3(CC3)C(N)=O)n2)cc1

InChI Key InChIKey=QCOBLDQZJWXXDC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 202418   

TargetVascular endothelial growth factor receptor 2(Human)
Cancer Therapeutics Crc Pty

US Patent
LigandPNGBDBM202418(US9238644, 24A)
Affinity DataIC50: 209nMpH: 7.2 T: 2°CAssay Description:Adult human umbilical vein endothelial cells (HUVEC) (Cat# CC-2519, Lonza) were seeded into clear-bottom, TC treated 12 well plates (Cat #665180, Gre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2016
Entry Details
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TargetVascular endothelial growth factor receptor 3(Human)
Cancer Therapeutics Crc Pty

US Patent
LigandPNGBDBM202418(US9238644, 24A)
Affinity DataIC50: 14nMpH: 7.4Assay Description:A biotin labelled peptide is used as substrate (amino acid sequence: Biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2)....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2016
Entry Details
Go to US Patent