BDBM200983 4,6-dimethyl-5-[2-methyl-4-(1,6-naphthyridin- 5-yloxy)phenyl]pyridazin-3(2H)-one::US9540352, example 10

SMILES Cc1cc(Oc2nccc3ncccc23)ccc1-c1c(C)n[nH]c(=O)c1C

InChI Key InChIKey=PQNZWZFBDINNSR-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 200983   

TargetD(1A) dopamine receptor(Human)
Pfizer

US Patent
LigandPNGBDBM200983(US9540352, example 10 | 4,6-dimethyl-5-[2-methyl-4...)
Affinity DataKi:  124nMpH: 7.4Assay Description:The affinity of the compounds described herein was determined by competition binding assays similar to those described in Ryman-Rasmussen et al., Dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2018
Entry Details
Go to US Patent