BDBM200822 8-hydroxy-2-[2-methyl-6-((2s,3'r)-2-methyl-[1,3']bipyrrolidinyl-1'-yl)-pyridin-3-yl]-2-aza-spiro[4.5]decan-1-one::US9533995, 5

SMILES C[C@H]1CCCN1[C@@H]1CCN(C1)c1ccc(N2CCC3(CCC(O)CC3)C2=O)c(C)n1

InChI Key InChIKey=AZBQFBWFMZCYJD-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 200822   

TargetHistamine receptor H3(Rhesus macaque)
Sanofi

US Patent
LigandPNGBDBM200822(8-hydroxy-2-[2-methyl-6-((2s,3'r)-2-methyl-[1,...)
Affinity DataKi:  267nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
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