BDBM200523 US9227970, 25

SMILES COc1ncc(nc1C(=O)Nc1ccc2nc(nn2c1)-c1ccccc1)C1CC1

InChI Key InChIKey=QPFCQEDSBRPEHH-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 200523   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Hoffmann-La Roche

US Patent

LigandBDBM200523(US9227970, 25)Copy SMILESCopy InChI

Affinity DataIC50: 17nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 ul contained 20 mM HEPES pH=7.5/10 mM MgCl...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
11/14/2016
Entry Details
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