BDBM200519 US9227970, 21

SMILES CN(C)c1nc2ccc(NC(=O)c3c(cnn3C)C(=O)N3CCCC3)cn2n1

InChI Key InChIKey=BFHHRKYKYJJHAB-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 200519   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Hoffmann-La Roche

US Patent

LigandBDBM200519(US9227970, 21)Copy SMILESCopy InChI

Affinity DataIC50: 28.6nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 ul contained 20 mM HEPES pH=7.5/10 mM MgCl...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
11/14/2016
Entry Details
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