BDBM197731 US9216986, 2-[(Z)-2-(5,7-Dimethyl-imidazo[1,2-a]pyrimidin-2-yl)-vinyl]-quinoline::US9801878, 2-[(Z)-2-(5,7-Dimethyl-imidazo[1,2-a]pyrimidin-2-yl)-vinyl]-quinoline

SMILES Cc1cc(C)n2cc(\C=C/c3ccc4ccccc4n3)nc2n1

InChI Key InChIKey=VCJQMIGZVTVBKJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 197731   

LigandPNGBDBM197731(US9216986, 2-[(Z)-2-(5,7-Dimethyl-imidazo[1,2-a]py...)
Affinity DataIC50: 240nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
Go to US Patent

LigandPNGBDBM197731(US9216986, 2-[(Z)-2-(5,7-Dimethyl-imidazo[1,2-a]py...)
Affinity DataIC50: 240nMAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2019
Entry Details
Go to US Patent