BDBM196938 US9212196, Derivative 34

SMILES COc1cc(CP(O)(=O)CC[C@@H](N)C(O)=O)cc(F)c1OCC(O)=O

InChI Key InChIKey=HLWOFNYCURCWQU-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 196938   

TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Descartes

US Patent
LigandPNGBDBM196938(US9212196, Derivative 34)
Affinity DataEC50:  3.09E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
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TargetMetabotropic glutamate receptor 8(Rat)
Universite Paris Descartes

US Patent
LigandPNGBDBM196938(US9212196, Derivative 34)
Affinity DataEC50:  9.17E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
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TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Descartes

US Patent
LigandPNGBDBM196938(US9212196, Derivative 34)
Affinity DataEC50:  2.32E+5nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
Go to US Patent