BDBM196652 US10329280, Compound I-2::US9212145, I-2

SMILES Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3nnc(N)n23)c1

InChI Key InChIKey=HNCMVNMHWKJIJY-UHFFFAOYSA-N

Data  2 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 196652   

TargetVascular endothelial growth factor receptor 2(Human)
Kala Pharmaceuticals

US Patent
LigandPNGBDBM196652(US9212145, I-2 | US10329280, Compound I-2)
Affinity DataKd:  2.80E+3nMAssay Description:A competition binding assay (DiscoveRx KINOMEscan) was used to measure the ability of the compound to compete for binding of an immobilized adenosine...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
Go to US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Kala Pharmaceuticals

US Patent
LigandPNGBDBM196652(US9212145, I-2 | US10329280, Compound I-2)
Affinity DataKd:  2.80E+3nMAssay Description:A competition binding assay (DiscoveRx KINOMEscan ) was used to measure the ability of the compound to compete for binding of an immobilized adenosin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/11/2020
Entry Details
Go to US Patent