BDBM192897 US9193689, IQ-080

SMILES CN1CCN(Cc2ccc(cc2)-c2cc3c(C)cc(F)cc3c(=O)[nH]2)CC1

InChI Key InChIKey=AKGKAUQMOQCXDE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 192897   

TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Human)
Institute of Cancer Research

US Patent
LigandPNGBDBM192897(US9193689, IQ-080)
Affinity DataIC50: 29nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2016
Entry Details
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