BDBM192295 US9187450, 43::US9321747, 12

SMILES CC(C)(O)CCOc1cnc(nc1)N1CCC(CC1)c1nc2CC(C)(C)C[C@H](O)c2c(C2CCC(F)(F)CC2)c1[C@@H](F)c1ccc(cc1)C(F)(F)F

InChI Key InChIKey=XVUDQBUEUFZZQH-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 192295   

TargetCholesteryl ester transfer protein(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM192295(US9187450, 43 | US9321747, 12)
Affinity DataIC50: 9nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 ug) and 5,5'-d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2016
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM192295(US9187450, 43 | US9321747, 12)
Affinity DataIC50: 17.8nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM192295(US9187450, 43 | US9321747, 12)
Affinity DataIC50: 21.3nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM192295(US9187450, 43 | US9321747, 12)
Affinity DataIC50: 22.7nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM192295(US9187450, 43 | US9321747, 12)
Affinity DataIC50: 11.6nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM192295(US9187450, 43 | US9321747, 12)
Affinity DataIC50: 13nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM192295(US9187450, 43 | US9321747, 12)
Affinity DataIC50: 28.9nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2017
Entry Details
Go to US Patent

TargetCholesteryl ester transfer protein(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM192295(US9187450, 43 | US9321747, 12)
Affinity DataIC50: 27.8nMT: 2°CAssay Description:A recombinant human CETP protein (manufactured by Roar Biomedical Inc.; 4.5 ng), the acceptor lipoprotein described in (2) above (32.5 μg) and 5,5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2017
Entry Details
Go to US Patent