BDBM163221 US9062045, 61

SMILES Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncc(cc4c3)N3CCC(F)(F)CC3)n2c1

InChI Key InChIKey=OHQMOXPQJBEGOZ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 163221   

LigandPNGBDBM163221(US9062045, 61)
Affinity DataIC50: 1.20E+4nMAssay Description:The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2016
Entry Details
Go to US Patent

TargetHepatocyte growth factor receptor(Human)
Novartis

US Patent
LigandPNGBDBM163221(US9062045, 61)
Affinity DataIC50: 4nMAssay Description:The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2016
Entry Details
Go to US Patent