BDBM159590 US9034921, E233

SMILES OC[C@H]1O[C@H]([C@H](O)[C@@H](O)[C@@H]1O)c1cc(Cc2ccc(cc2)C2CCCC2)c(Cl)c2OCCc12

InChI Key InChIKey=DDNVQOAZSNCRND-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 159590   

TargetSodium/glucose cotransporter 2(Human)
Green Cross

US Patent
LigandPNGBDBM159590(US9034921, E233)
Affinity DataIC50: 1.16nMpH: 7.4 T: 2°CAssay Description:For sodium-dependent glucose transport assay, cells expressing hSGLT2 were seeded into a 96-well culture plate at a density of 5x104 cells/well in RP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2015
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 2(Human)
Green Cross

US Patent
LigandPNGBDBM159590(US9034921, E233)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetSodium/glucose cotransporter 1(Human)
Gc Pharma

Curated by ChEMBL
LigandPNGBDBM159590(US9034921, E233)
Affinity DataIC50: 9.93E+3nMAssay Description:Inhibition of human SGLT1 expressed in CHO cells by methyl-alpha-D-glucopyranoside assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed