BDBM159401 US9034921, E017::US9340521, E011

SMILES CCc1ccc(Cc2cc([C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c3OCCCc3c2Cl)cc1

InChI Key InChIKey=PFKDLBHFBULNCB-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 159401   

TargetSodium/glucose cotransporter 2(Human)
Green Cross

US Patent
LigandPNGBDBM159401(US9034921, E017 | US9340521, E011)
Affinity DataIC50: 0.845nMpH: 7.4 T: 2°CAssay Description:For sodium-dependent glucose transport assay, cells expressing hSGLT2 were seeded into a 96-well culture plate at a density of 5x104 cells/well in RP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2015
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Green Cross

US Patent
LigandPNGBDBM159401(US9034921, E017 | US9340521, E011)
Affinity DataIC50: 0.850nMpH: 7.4 T: 2°CAssay Description:For sodium-dependent glucose transport assay, cells expressing hSGLT2 were seeded into a 96-well culture plate at a density of 5×104 cells/well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Green Cross

US Patent
LigandPNGBDBM159401(US9034921, E017 | US9340521, E011)
Affinity DataIC50: 27nMpH: 7.4 T: 2°CAssay Description:For sodium-dependent glucose transport assay, cells expressing hSGLT1 were seeded into a 96-well culture plate at a density of 5×104 cells/well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2017
Entry Details
Go to US Patent