BDBM155363 US10383871, Example 9::US10918640, Example 9::US9006269, 9

SMILES O=C(Nc1cccnn1)N1CC(C1)Oc1ccc(cn1)-c1cccc(OCCOCc2ccccc2)c1

InChI Key InChIKey=KWGBRFMUYCLMJO-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 155363   

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155363(US9006269, 9 | US10383871, Example 9 | US10918640,...)
Affinity DataIC50: 3nMpH: 8.2 T: 2°CAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2015
Entry Details
Go to US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155363(US9006269, 9 | US10383871, Example 9 | US10918640,...)
Affinity DataIC50: 3nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2020
Entry Details
Go to US Patent

TargetFatty-acid amide hydrolase 1(Human)
Vernalis (R&D)

US Patent
LigandPNGBDBM155363(US9006269, 9 | US10383871, Example 9 | US10918640,...)
Affinity DataIC50: 3nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
Go to US Patent