BDBM151750 BDBM151751::US8987445, 186

SMILES OC(=O)c1ccc(cc1)S(=O)(=O)N(C1CCc2cc(OC(F)(F)F)ccc12)c1ncc2ccccc2c1C1CC1

InChI Key InChIKey=RLONLJJPXIVWOF-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 151750   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM151750(BDBM151751 | US8987445, 186)
Affinity DataIC50: 4.30nMT: 2°CAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+ sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
Go to US Patent

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM151750(BDBM151751 | US8987445, 186)
Affinity DataIC50: 128nMT: 2°CAssay Description:The functional activity of compounds was determined by measuring changes in intracellular calcium concentration using a Ca2+ sensitive fluorescent dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
Go to US Patent