BDBM150751 CPR005231 (6)

SMILES COc1cc(ccc1O)-c1ccc2ccc(-c3cccc(c3)C(=O)NCCN(C)C)n2n1

InChI Key InChIKey=MCIDHQCNUZBVQJ-UHFFFAOYSA-N

Data  5 IC50  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 150751   

TargetDeath-associated protein kinase 1(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 247nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataKd:  240nMpH: 7.5Assay Description:40 µL of a solution containing 350-500 µM of CPR005231 (compound 6) were titrated into the 200 µL sample cell containing 25-55 µM DAPK1 (AA 1-285) or...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 1.60E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 1.80E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 5(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 5.60E+3nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Copenhagen

LigandPNGBDBM150751(CPR005231 (6))
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:The reaction was started by adding a mix of ATP and Peptide 38 to assay plates containing DAPK1. Prior to mixing, all reagents are diluted in assay b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2015
Entry Details Article
PubMed