BDBM149202 US8962648, 1324

SMILES C[C@@H](CN(C)C)c1ccc(cc1)-c1c(O)cc(C)c2[nH]c(=O)c3sccc3c12

InChI Key InChIKey=XCFRUAOZMVFDPQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 149202   

TargetLymphokine-activated killer T-cell-originated protein kinase(Human)
Oncotherapy Science

US Patent
LigandPNGBDBM149202(US8962648, 1324)
Affinity DataIC50: 32nMpH: 7.4 T: 2°CAssay Description:PBK activity was determined in the presence or absence of compounds using fluorescein isothiocyanate-labeled (FITC-labeled) histone H3 peptide as a s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2015
Entry Details
Go to US Patent

TargetLymphokine-activated killer T-cell-originated protein kinase(Human)
Oncotherapy Science

US Patent
LigandPNGBDBM149202(US8962648, 1324)
Affinity DataIC50: 354nMAssay Description:Inhibition of human TOPK using MBP as substrate after 2 hrs in presence of [gamma-33P]-ATP by filter-binding methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed