BDBM148095 US8962609, DMX-27

SMILES Cn1nccc1Nc1nccc(n1)-c1ccc(N2CCCC2)c(c1)C#N

InChI Key InChIKey=DAZUIYGZOWVNPV-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 148095   

TargetSerine/threonine-protein kinase TBK1(Human)
Domainex

US Patent
LigandPNGBDBM148095(US8962609, DMX-27)
Affinity DataIC50: 30nMpH: 7.5Assay Description:Inhibitions studies were performed using a time-resolved fluorescence-based Lanthascreen assay. Phosphorylation of a fluorescein-labelled substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent

LigandPNGBDBM148095(US8962609, DMX-27)
Affinity DataIC50: 300nMpH: 7.5Assay Description:Inhibitions studies were performed using a time-resolved fluorescence-based Lanthascreen assay. Phosphorylation of a fluorescein-labelled substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2015
Entry Details
US Patent