BDBM146685 US8957073, 4.19::US9718803, 4.19

SMILES Cc1cncc(c1)-c1nccnc1C1CN(C1)c1ccc2ccccc2n1

InChI Key InChIKey=PBLYFTOVXAUJDE-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 146685   

LigandPNGBDBM146685(US8957073, 4.19 | US9718803, 4.19)
Affinity DataIC50: 0.0163nMT: 2°CAssay Description:Enzyme Activity. An IMAP TR-FRET assay was used to analyze the enzyme activity (Molecular Devices Corp., Sunnyvale Calif.). 5 uL of serial diluted PD...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2015
Entry Details
Go to US Patent

LigandPNGBDBM146685(US8957073, 4.19 | US9718803, 4.19)
Affinity DataIC50: 0.0160nMT: 2°CAssay Description:An IMAP TR-FRET assay was used to analyze the enzyme activity (Molecular Devices Corp., Sunnyvale Calif.). 5 L of serial diluted PDE10A (BPS Bioscien...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2018
Entry Details
Go to US Patent