BDBM144682 US8952037, 55

SMILES N#Cc1ccc(cn1)-c1cccnc1O[C@@H]1C[C@@H](C1)Nc1ccc2ccccc2n1

InChI Key InChIKey=XOKPHIOYZUXZHP-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 144682   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Amgen

US Patent

LigandBDBM144682(US8952037, 55)Copy SMILESCopy InChI

Affinity DataIC50: 1.29nMT: 2°CAssay Description:Enzyme Activity. An IMAP TR-FRET assay was used to analyze the enzyme activity (Molecular Devices Corp., Sunnyvale Calif.). 5 uL, of serial diluted P...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
6/29/2015
Entry Details
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