BDBM144668 US8952037, 41

SMILES Clc1ccc(C2=CCOCC2)c(O[C@@H]2C[C@@H](C2)Nc2nc3ccccc3s2)n1

InChI Key InChIKey=XPRMRYWRDCTTSY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 144668   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Amgen

US Patent

LigandBDBM144668(US8952037, 41)Copy SMILESCopy InChI

Affinity DataIC50: 3.55nMT: 2°CAssay Description:Enzyme Activity. An IMAP TR-FRET assay was used to analyze the enzyme activity (Molecular Devices Corp., Sunnyvale Calif.). 5 uL, of serial diluted P...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
6/29/2015
Entry Details
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