BDBM142657 US8937068, 46

SMILES CCN(C(C)=O)C(=O)Nc1ccc2ncc(nc2n1)-c1ccccc1

InChI Key InChIKey=MRGFJFFONCTHQQ-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 142657   

TargetMitogen-activated protein kinase 1(Human)
Zentaris

US Patent
LigandPNGBDBM142657(US8937068, 46)
Affinity DataIC50: 9.50E+3nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
Go to US Patent

LigandPNGBDBM142657(US8937068, 46)
Affinity DataIC50: 1.00E+5nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 14(Human)
Zentaris

US Patent
LigandPNGBDBM142657(US8937068, 46)
Affinity DataIC50: 495nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 8/9(Human)
Zentaris

US Patent
LigandPNGBDBM142657(US8937068, 46)
Affinity DataIC50: 1.00E+5nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2015
Entry Details
Go to US Patent