BDBM141349 US8916594, I-029

SMILES CCS(=O)(=O)NC[C@H]1CC[C@@H](CC1)Nc1nc(no1)-c1ccc(F)c(F)c1

InChI Key InChIKey=UPBJWRXHQFMCET-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 141349   

TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM141349(US8916594, I-029)
Affinity DataIC50: 0.220nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2015
Entry Details
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TargetNeuropeptide Y receptor type 5(Human)
Shionogi

US Patent
LigandPNGBDBM141349(US8916594, I-029)
Affinity DataIC50: 0.860nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a human NPY Y5 receptor (WO96/16542) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Biol. 8, 466-472). The obtained ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2015
Entry Details
Go to US Patent