BDBM128022 US8796328, B::US8802711, I

SMILES CC(C)(C)c1ccc(Nc2ncnc3cc(ccc23)-c2ncccc2C(F)(F)F)cc1

InChI Key InChIKey=RXRYUCSWVNXEHU-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 128022   

LigandPNGBDBM128022(US8802711, I | US8796328, B)
Affinity DataIC50: 55nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2]i) using the Fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2014
Entry Details
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LigandPNGBDBM128022(US8802711, I | US8796328, B)
Affinity DataIC50: 55nMAssay Description:The functional activity of compounds at the TRPV1 receptor was determined by measurement of intracellular Ca2+ levels ([Ca2+]i) using the Fluorescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2015
Entry Details
Go to US Patent

LigandPNGBDBM128022(US8802711, I | US8796328, B)
Affinity DataIC50: 55nMAssay Description:The cDNA for human TRPV1 (hTRPV1) was isolated by reverse transcriptase-polymerase chain reaction (RT-PCR) from human small intestine poly A+ RNA sup...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
Go to US Patent