BDBM126129 US8779142, 153

SMILES Cn1cc(cn1)-c1cn(cn1)-c1ccnc2n(nc(c12)C(F)(F)F)-c1ccc(cc1Cl)C(N)=O

InChI Key InChIKey=GKUKNUORVOHZBH-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 126129   

TargetHeat shock protein HSP 90-alpha(Human)
Taiho Pharmaceutical

US Patent

LigandBDBM126129(US8779142, 153)Copy SMILESCopy InChI

Affinity DataIC50: 130nMpH: 7.5Assay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
12/8/2014
Entry Details
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