BDBM104264 CHEMBL1950750::US8575186, 27

SMILES Cn1c2CC3CCC(N3)c2c2cc(ccc12)S(=O)(=O)c1ccccc1

InChI Key InChIKey=LKNYHWXHAONTOU-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 104264   

Target5-hydroxytryptamine receptor 6(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104264(CHEMBL1950750 | US8575186, 27)
Affinity DataKi:  7.80nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 6(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104264(CHEMBL1950750 | US8575186, 27)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104264(CHEMBL1950750 | US8575186, 27)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104264(CHEMBL1950750 | US8575186, 27)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed