BDBM82251 (R)-4-Carboxyphenylglycine::(S)-4CPG::CAS_134052-68-9

SMILES N[C@@H](C(O)=O)c1ccc(cc1)C(O)=O

InChI Key InChIKey=VTMJKPGFERYGJF-UHFFFAOYSA-N

Data  10 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 82251   

TargetCystine/glutamate transporter(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of xc-cystine-glutamate antiporter-mediated cystine uptake in human U87 cells using L-[14C]cystine as substrate after 15 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi:  3.70E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetGlutamate receptor 3(Rat)
Novo Nordisk

Curated by PDSP Ki Database
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Novo Nordisk

Curated by PDSP Ki Database
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Novo Nordisk

Curated by PDSP Ki Database
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Novo Nordisk

Curated by PDSP Ki Database
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Novo Nordisk

Curated by PDSP Ki Database
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Novo Nordisk

Curated by PDSP Ki Database
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM82251((S)-4CPG | CAS_134052-68-9 | (R)-4-Carboxyphenylgl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed