BDBM20255 4-[(2S)-2-{[(1S,2R)-1-{[(1S)-2-carbamoyl-1-{[(1S)-3-carbamoyl-1-{[(1S)-1-{[(1S)-1-carbamoyl-2-methylpropyl]carbamoyl}-2-hydroxyethyl]carbamoyl}propyl]carbamoyl}ethyl]carbamoyl}-2-methylbutyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid::EGFR (1068) derived peptide, 11::Y(p)INQSV

SMILES CCC(C)[C@H](NC(=O)[C@H](Cc1ccc(OP(O)(O)=O)cc1)NC(C)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C(C)C)C(N)=O

InChI Key InChIKey=JRBFXEOBSAAIFI-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20255   

TargetSignal transducer and activator of transcription 3(Mouse)
The University of Texas At Houston

LigandPNGBDBM20255(Y(p)INQSV | 4-[(2S)-2-{[(1S,2R)-1-{[(1S)-2-carbamo...)
Affinity DataIC50: 3.00E+4nMpH: 7.8 T: 2°CAssay Description:His10-Stat3 was expressed in Sf9 cells from a baculovirus encoding the recombinant protein. A nuclear extract of the Sf9 cells was incubated with 32P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2008
Entry Details Article
PubMed