BDBM35343 indole-2-carboxamide derivative, 9b::trans-isomers+ 9a

SMILES O[C@H]1CCc2cc(NC(=O)c3cc4cc(Cl)ccc4[nH]3)ccc2[C@@H]1O

InChI Key InChIKey=OPIRGJRMKUMHMK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 35343   

TargetGlycogen phosphorylase, liver form(Human)
Astellas Pharma

LigandPNGBDBM35343(trans-isomers+ 9a | indole-2-carboxamide derivativ...)
Affinity DataIC50: 800nMpH: 6.8 T: 2°CAssay Description:The activity of recombinant human liver GPa in the forward direction was measured by monitoring the production of NADPH. Enzyme activity was assayed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2009
Entry Details Article
PubMed