BDBM62877 2-(2-ketopyrrolidino)acetamide::2-(2-oxidanylidenepyrrolidin-1-yl)ethanamide::2-(2-oxo-1-pyrrolidinyl)acetamide::2-(2-oxopyrrolidin-1-yl)acetamide::MLS000069719::PIRACETAM::SMR000058196::cid_4843

SMILES C1CC(=O)N(C1)CC(=O)N

InChI Key InChIKey=GMZVRMREEHBGGF-UHFFFAOYSA-N

Data  6 IC50  1 EC50

PDB links: 2 PDB IDs match this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 62877   

TargetHeat shock factor protein 1(Mouse)
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM62877(2-(2-oxopyrrolidin-1-yl)acetamide | PIRACETAM | ci...)
Affinity DataEC50: >1.95E+5nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2011
Entry Details
PCBioAssay
TargetSynaptic vesicle glycoprotein 2A(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM62877(2-(2-oxopyrrolidin-1-yl)acetamide | PIRACETAM | ci...)
Affinity DataIC50: 3.98E+4nMAssay Description:In vitro inhibitory activity against [3H](2S)-2-[4-(3-azidophenyl)-2-oxopyrrolidin-1-yl]butanamide binding to levetiracetam binding siteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBile salt export pump(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM62877(2-(2-oxopyrrolidin-1-yl)acetamide | PIRACETAM | ci...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human BSEP expressed in baculovirus transfected fall armyworm Sf21 cell membranes vesicles assessed as reduction in ATP-dependent [3H]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2019
Entry Details Article
PubMed
LigandPNGBDBM62877(2-(2-oxopyrrolidin-1-yl)acetamide | PIRACETAM | ci...)
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human MRP2 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMed
LigandPNGBDBM62877(2-(2-oxopyrrolidin-1-yl)acetamide | PIRACETAM | ci...)
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human MRP3 overexpressed in Sf9 insect cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMed
LigandPNGBDBM62877(2-(2-oxopyrrolidin-1-yl)acetamide | PIRACETAM | ci...)
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMed
TargetBile salt export pump(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM62877(2-(2-oxopyrrolidin-1-yl)acetamide | PIRACETAM | ci...)
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMed