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21 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Inhibitors of Influenza Virus Polymerase Acidic (PA) Endonuclease: Contemporary Developments and Perspectives.EBI
Shandong University
Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Protein-Protein Interaction as a Target for Next-Generation Anti-influenza Therapeutics.EBI
University of Perugia
Virtual Screening and Biological Validation of Novel Influenza Virus PA Endonuclease Inhibitors.EBI
University of Sassari
Structural and computational study on inhibitory compounds for endonuclease activity of influenza virus polymerase.EBI
Chiba University
Inhibition of cap (m7GpppXm)-dependent endonuclease of influenza virus by 4-substituted 2,4-dioxobutanoic acid compounds.EBI
Merck Research Laboratories
Synthesis of natural flutimide and analogous fully substituted pyrazine-2,6-diones, endonuclease inhibitors of influenza virus.EBI
Merck Research Laboratories
Anti-influenza virus activities of 4-substituted 2,4-dioxobutanoic acid inhibitors.EBI
Merck Research Laboratories
Identification of influenza endonuclease inhibitors using a novel fluorescence polarization assay.EBI
University of Tennessee Health Science Center
Tetramic and tetronic acids: an update on new derivatives and biological aspects.EBI
University of Bayreuth
Bioisosteres of the Phenyl Ring: Recent Strategic Applications in Lead Optimization and Drug Design.EBI
Biocon-Bristol Myers Squibb Research and Development Centre
Geminal Diheteroatomic Motifs: Some Applications of Acetals, Ketals, and Their Sulfur and Nitrogen Homologues in Medicinal Chemistry and Drug Design.EBI
Bristol Myers Squibb Research and Early Development
Discovery and optimization of new 6, 7-dihydroxy-1, 2, 3, 4-tetrahydroisoquinoline derivatives as potent influenza virus PAEBI
South China Agricultural University
Use of a pharmacophore model to discover a new class of influenza endonuclease inhibitors.EBI
Roche Discovery Welwyn
Fragment-Based Identification of Influenza Endonuclease Inhibitors.EBI
University of California San Diego
SAR Exploration of Tight-Binding Inhibitors of Influenza Virus PA Endonuclease.EBI
University of California
Synthesis and SAR Study of Carbamoyl Pyridone Bicycle Derivatives as Potent Inhibitors of Influenza Cap-dependent Endonuclease.EBI
Shionogi
Non-chelating p-phenylidene-linked bis-imidazoline analogs of known influenza virus endonuclease inhibitors: Synthesis and anti-influenza activity.EBI
Saint Petersburg State University
Identification of N- and C-3-Modified Laudanosoline Derivatives as Novel Influenza PAEBI
South China Agricultural University
Identification of influenza PA-Nter endonuclease inhibitors using pharmacophore- and docking-based virtual screening.EBI
Polo Universitario Ss. Annunziata
Quinoline analogs as phosphatidylinositol 3-kinase inhibitorsBDB
Nanjing Zhengxiang Pharmaceuticals
WDR5 inhibitors and modulatorsBDB
Vanderbilt University